SCHEMBL8024017

SCHEMBL8024017

Clc1cccc(Nc2ccc(-c3ccccc3)nn2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.61
ALDH1A1 P00352 3/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
ABCG2 Q9UNQ0 2/20 0.53
ABCB1 P08183 1/20 0.53
ABCC1 P33527 1/20 0.53
PDE5A O76074 3/20 0.51
MAPT P10636 3/20 0.51
KDM4E B2RXH2 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
HPGD P15428 1/20 0.51
ALOX15 P16050 1/20 0.51
CYP2C19 P33261 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28706653 0.87 MEN1 (0.57) DGAT1ALDH1A1MEN1KMT2ANPC1
SCHEMBL180521 0.85 DGAT1 (0.71) DGAT1ALDH1A1MEN1KMT2ANPC1
SCHEMBL1752922 0.84 RAB9A (0.62) DGAT1ALDH1A1MEN1KMT2ANPC1
SCHEMBL12203212 0.80 DGAT1 (0.51) DGAT1ALDH1A1MEN1KMT2ANPC1
SCHEMBL29818154 0.79 ALDH1A1 (0.54) DGAT1ALDH1A1MEN1KMT2ANPC1
SCHEMBL3595694 0.79 ALDH1A1 (0.68) DGAT1ALDH1A1MEN1KMT2AABCG2
SCHEMBL31592780 0.79 ALDH1A1 (0.58) DGAT1ALDH1A1MEN1KMT2ANPC1
SCHEMBL2300032 0.78 MEN1 (0.75) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL3580458 0.78 HTR3E (0.53) DGAT1ALDH1A1MEN1KMT2AABCG2
SCHEMBL8011183 0.77 MAPT (0.55) DGAT1ALDH1A1MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0975605-A1 PYRIDAZINE AND PHTHALAZINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-02-02 EP claimed
WO-1998046574-A1 PYRIDAZINE AND PHTHALAZINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1998-10-22 WO claimed
EP-0975605-A1 PYRIDAZINE AND PHTHALAZINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 2000-02-02 EP disclosed
WO-1998046574-A1 PYRIDAZINE AND PHTHALAZINE DERIVATIVES, PROCESS OF THEIR PREPARATION AND THEIR USE AS ANTICONVULSANTS SMITHKLINE BEECHAM PLC (GB) 1998-10-22 WO disclosed