SCHEMBL8025317

SCHEMBL8025317

CCOc1ccc(N2CCc3ccccc3C2)c2cccnc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.51
LMNA P02545 5/20 0.48
GAA P10253 4/20 0.48
HTT P42858 5/20 0.47
POLB P06746 2/20 0.47
MAPT P10636 6/20 0.47
KDM4E B2RXH2 3/20 0.47
NPSR1 Q6W5P4 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
MAPK1 P28482 1/20 0.47
NUDT1 P36639 1/20 0.46
GRIN2D O15399 2/20 0.45
GRIN3B O60391 2/20 0.45
GRIN1 Q05586 2/20 0.45
GRIN2A Q12879 2/20 0.45
GRIN2B Q13224 2/20 0.45
GRIN2C Q14957 2/20 0.45
GRIN3A Q8TCU5 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
ALOX12 P18054 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6160557 0.78 NUDT1 (0.52) ALDH1A1MAPTKDM4ENPSR1L3MBTL1
Hydrochloric Acid SCHEMBL6161091 0.71 NUDT1 (0.55) LMNAHTTPOLBMAPTKDM4E
SCHEMBL6159581 0.69 NUDT1 (0.63) LMNAMAPTNUDT1GRIN2DGRIN3B
Hydrochloric Acid SCHEMBL6162260 0.68 NUDT1 (0.61) LMNAMAPTNUDT1GRIN2DGRIN3B
SCHEMBL18029399 0.68 PSMD14 (0.59) ALDH1A1LMNAHTTPOLBMAPT
SCHEMBL8035380 0.67 LMNA (0.44) ALDH1A1LMNAGAAHTTPOLB
SCHEMBL10094645 0.67 GRIN2D (0.68) ALDH1A1LMNAHTTGRIN2DGRIN3B
SCHEMBL23359957 0.67 ALDH1A1 (0.51) ALDH1A1LMNAGAAHTTPOLB
SCHEMBL10650819 0.67 PKM (0.62) ALDH1A1LMNAGAAHTTPOLB
SCHEMBL28169008 0.67 ALDH1A1 (0.49) ALDH1A1LMNAGAAHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993449-A1 QUINOLINE DERIVATIVES AS PDE IV AND/OR TNF INHIBITORS Darwin Discovery Limited (GB) 2000-04-19 EP claimed
WO-1998057936-A1 QUINOLINE DERIVATIVES AS PDE IV AND/OR TNF INHIBITORS DARWIN DISCOVERY LIMITED (GB) 1998-12-23 WO claimed
US-6069151-A Quinolines and their therapeutic use DARWIN DISCOVERY, LTD. (GB) 2000-05-30 US disclosed