SCHEMBL8025473

SCHEMBL8025473

COc1cc(Cl)c(C(=O)N(C)C(=O)N(C(C)C)C(C)C)cc1O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPT P10636 3/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
NPC1 O15118 1/20 0.37
MAPK1 P28482 1/20 0.37
NOD2 Q9HC29 1/20 0.37
HPGD P15428 3/20 0.36
LMNA P02545 1/20 0.36
CYP3A4 P08684 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
CXCL12 P48061 3/20 0.35
ALDH1A1 P00352 2/20 0.35
STAT3 P40763 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025474 0.82 TSHR (0.39) HSP90AA1KDM4EMAPTMEN1KMT2A
SCHEMBL8035585 0.81 HSP90AA1 (0.41) HSP90AA1KDM4EMAPTHPGDLMNA
SCHEMBL8039002 0.81 MAPT (0.39) HSP90AA1KDM4EMAPTMEN1KMT2A
SCHEMBL8035119 0.78 KDM4E (0.40) HSP90AA1KDM4EMAPTMEN1KMT2A
SCHEMBL8039019 0.78 HSP90AA1 (0.39) HSP90AA1KDM4EMAPTMEN1KMT2A
SCHEMBL8031650 0.77 MEN1 (0.46) MEN1KMT2ANPC1HPGDHTT
SCHEMBL8039011 0.77 HSP90AA1 (0.53) HSP90AA1KDM4EMAPTMEN1KMT2A
SCHEMBL8039013 0.76 ALDH1A1 (0.41) HSP90AA1MEN1KMT2AHPGDLMNA
SCHEMBL8032092 0.76 ALDH1A1 (0.44) KDM4EMAPTMEN1KMT2ANPC1
SCHEMBL8039016 0.75 HTT (0.42) HSP90AA1KDM4ELMNAHTTCXCL12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed