SCHEMBL8025474

SCHEMBL8025474

COc1cc(Cl)c(C(=O)N(C)C(=O)N(C)C2CC2)cc1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.39
HPGD P15428 2/20 0.39
HSP90AA1 P07900 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
NPC1 O15118 1/20 0.36
MAPK1 P28482 1/20 0.36
NOD2 Q9HC29 1/20 0.36
LMNA P02545 2/20 0.35
CYP3A4 P08684 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35
DRD1 P21728 2/20 0.34
DRD5 P21918 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LPAR5 Q9H1C0 1/20 0.34
MAOA P21397 2/20 0.34
CXCL12 P48061 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025473 0.82 HSP90AA1 (0.37) TSHRHPGDHSP90AA1MEN1KMT2A
SCHEMBL8032092 0.79 ALDH1A1 (0.44) TSHRHPGDMEN1KMT2AKDM4E
SCHEMBL8035585 0.79 HSP90AA1 (0.41) TSHRHPGDHSP90AA1KDM4EMAPT
SCHEMBL8022338 0.78 TRPM8 (0.46) HPGDMEN1KMT2ANPC1
SCHEMBL8038341 0.78 SMO (0.38) TSHRHPGDMEN1KMT2AKDM4E
SCHEMBL8035119 0.76 KDM4E (0.40) HPGDHSP90AA1MEN1KMT2AKDM4E
SCHEMBL8039019 0.76 HSP90AA1 (0.39) TSHRHSP90AA1MEN1KMT2AKDM4E
SCHEMBL8039011 0.75 HSP90AA1 (0.53) TSHRHPGDHSP90AA1MEN1KMT2A
SCHEMBL8039013 0.74 ALDH1A1 (0.41) TSHRHPGDHSP90AA1MEN1KMT2A
SCHEMBL8041629 0.74 TDP1 (0.34) TSHRHPGDMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed