SCHEMBL8025972

SCHEMBL8025972

Cc1cc2c(C(CO)N3CCCC[C@H]3C)cccc2n1C

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 4/20 0.36
NPSR1 Q6W5P4 2/20 0.36
P2RX7 Q99572 1/20 0.35
CHRM2 P08172 1/20 0.34
HSD17B10 Q99714 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH3 Q9Y5N1 4/20 0.32
TSHR P16473 3/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.31
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
SYK P43405 1/20 0.31
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7210503 0.69 KDM4E (0.37) KDM4EALDH1A1NPSR1P2RX7MEN1
SCHEMBL7210500 0.69 KDM4E (0.37) KDM4EALDH1A1NPSR1P2RX7MEN1
Hydrochloric Acid SCHEMBL7210309 0.68 KDM4E (0.39) KDM4EALDH1A1NPSR1P2RX7MEN1
SCHEMBL8015495 0.66 CYP1A2 (0.34) HSD17B10TSHR
SCHEMBL16202643 0.66 CASP1 (0.39) KDM4EHSD17B10MAPTTSHRHPGD
SCHEMBL5347104 0.66 KDM4E (0.54) KDM4EALDH1A1HRH3
SCHEMBL18000121 0.61 SLC6A4 (0.38) KDM4EHSD17B10SYK
SCHEMBL22434745 0.60 NPEPPS (0.46) KDM4EALDH1A1NPSR1HSD17B10MEN1
SCHEMBL18000284 0.60 MAPT (0.46) KDM4EALDH1A1HSD17B10MEN1MAPT
SCHEMBL13548554 0.59 ALKBH5 (0.52) KDM4EALDH1A1HSD17B10MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061554-A1 1-AMINO ETHYLINDOLE DERIVATIVES FOR THE TREATMENT OF URINARY INCONTINENCE SANOFI-SYNTHELABO (FR) 2000-10-19 WO claimed
WO-2000061554-A1 1-AMINO ETHYLINDOLE DERIVATIVES FOR THE TREATMENT OF URINARY INCONTINENCE SANOFI-SYNTHELABO (FR) 2000-10-19 WO disclosed