SCHEMBL8026786

SCHEMBL8026786

COC(=O)CN(C(=O)[C@@H](CCc1ccccc1)CSC(C)=O)c1cccc(OCc2ccc(C(=O)OC)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 3/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
MAOB P27338 1/20 0.38
CHRM3 P20309 3/20 0.38
POLB P06746 1/20 0.38
ALOX5 P09917 2/20 0.38
EPOR P19235 1/20 0.37
MRGPRX4 Q96LA9 1/20 0.37
PTGES O14684 1/20 0.37
LTC4S Q16873 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8020677 0.94 ALDH1A1 (0.43) ALDH1A1MAOBALOX5EPORPTGES
SCHEMBL8026727 0.94 MRGPRX4 (0.45) LNPEPSMN1; SMN2ALDH1A1MAOBMRGPRX4
SCHEMBL8026201 0.92 ALDH1A1 (0.46) LNPEPMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL8171062 0.88 MLYCD (0.41) ALDH1A1
SCHEMBL8026900 0.87 MRGPRX4 (0.46) LNPEPSMN1; SMN2ALDH1A1MRGPRX4
SCHEMBL8010485 0.86 ALDH1A1 (0.50) ALDH1A1MAOBALOX5EPOR
SCHEMBL8020308 0.86 MLYCD (0.41) PTGES
SCHEMBL8020571 0.86 ALDH1A1 (0.51) SMN1; SMN2ALDH1A1MAOBEPOR
SCHEMBL8010570 0.84 ALDH1A1 (0.48) MEN1KMT2AALDH1A1MAOB
SCHEMBL8022286 0.84 MLYCD (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed