SCHEMBL8020308

SCHEMBL8020308

COC(=O)CN(C(=O)C(CCc1ccccc1)CSC(C)=O)c1cccc(Oc2ccccc2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.41
CETP P11597 2/20 0.38
PTGES O14684 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
ABCC3 O15438 1/20 0.37
NR1I2 O75469 1/20 0.37
ABCB11 O95342 1/20 0.37
NR3C1 P04150 1/20 0.37
RARG P13631 1/20 0.37
CNR1 P21554 1/20 0.37
OPRK1 P41145 1/20 0.37
NR1H2 P55055 1/20 0.37
PPARA Q07869 1/20 0.37
NR1H3 Q13133 1/20 0.37
NR1I3 Q14994 1/20 0.37
FFAR1 O14842 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026202 0.96 MLYCD (0.39) MLYCDCETPOPRM1MTNR1AMTNR1B
SCHEMBL8020677 0.91 ALDH1A1 (0.43) MLYCDPTGESCYP1A2CYP3A4CYP2D6
SCHEMBL8020337 0.89 MLYCD (0.41) MLYCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8022286 0.89 MLYCD (0.41) MLYCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8022500 0.86 ALDH1A1 (0.40) MLYCDMTNR1AMTNR1B
SCHEMBL8026727 0.86 MRGPRX4 (0.45) CETP
SCHEMBL8026786 0.86 LNPEP (0.41) PTGES
SCHEMBL8023152 0.85 MLYCD (0.38) MLYCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8024569 0.84 MLYCD (0.45) MLYCDCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8010673 0.84 TSPO (0.44) MLYCDCYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed
EP-0934262-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1999-08-11 EP disclosed
WO-1998017639-A1 BETA-THIOPROPIONYL-AMINO ACID DERIVATIVES AND THEIR USE AS BETA-LACTAMASE INHIBITORS SMITHKLINE BEECHAM PLC (GB) 1998-04-30 WO disclosed