SCHEMBL8026727

SCHEMBL8026727

COC(=O)CN(C(=O)[C@@H](CCc1ccccc1)CSC(C)=O)c1cccc(OCc2cccc(C(=O)OC)c2)c1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 5/20 0.45
CETP P11597 1/20 0.39
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
MAOB P27338 1/20 0.38
LNPEP Q9UIQ6 1/20 0.38
ADAMTS4 O75173 1/20 0.37
MMP13 P45452 1/20 0.37
NR4A2 P43354 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026786 0.94 LNPEP (0.41) MRGPRX4ALDH1A1SMN1; SMN2MAOBLNPEP
SCHEMBL8026900 0.94 MRGPRX4 (0.46) MRGPRX4ALDH1A1KDM4EMAPTRAB9A
SCHEMBL8020677 0.93 ALDH1A1 (0.43) ALDH1A1MAOB
SCHEMBL8020308 0.86 MLYCD (0.41) CETP
SCHEMBL8026201 0.85 ALDH1A1 (0.46) ALDH1A1MAPTRAB9ASMN1; SMN2MAOB
SCHEMBL8020571 0.84 ALDH1A1 (0.51) ALDH1A1RAB9ASMN1; SMN2MAOB
SCHEMBL8022286 0.84 MLYCD (0.41) ALDH1A1
SCHEMBL8010485 0.83 ALDH1A1 (0.50) ALDH1A1MAOB
SCHEMBL8019970 0.83 ALDH1A1 (0.43) ALDH1A1MAOBLNPEP
SCHEMBL8171062 0.83 MLYCD (0.41) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed