SCHEMBL8020677

SCHEMBL8020677

COC(=O)CN(C(=O)C(CCc1ccccc1)CSC(C)=O)c1cccc(OCc2ccccc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
ALOX5 P09917 1/20 0.41
EPOR P19235 1/20 0.41
MAOB P27338 1/20 0.40
CYP2D6 P10635 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ABCC3 O15438 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
NR3C1 P04150 1/20 0.40
RARG P13631 1/20 0.40
CNR1 P21554 1/20 0.40
OPRK1 P41145 1/20 0.40
NR1H2 P55055 1/20 0.40
PPARA Q07869 1/20 0.40
NR1H3 Q13133 1/20 0.40
NR1I3 Q14994 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8026786 0.94 LNPEP (0.41) ALDH1A1ALOX5EPORMAOBPTGES
SCHEMBL8026727 0.93 MRGPRX4 (0.45) ALDH1A1MAOB
SCHEMBL8020308 0.91 MLYCD (0.41) CYP2D6CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8020571 0.91 ALDH1A1 (0.51) ALDH1A1EPORMAOBCYP2D6CYP1A2
SCHEMBL8010485 0.90 ALDH1A1 (0.50) ALDH1A1ALOX5EPORMAOBCYP2D6
SCHEMBL8022286 0.89 MLYCD (0.41) ALDH1A1CYP2D6CYP1A2CYP3A4CYP2C9
SCHEMBL8026202 0.88 MLYCD (0.39) ALDH1A1MLYCDMTNR1AMTNR1B
SCHEMBL8010570 0.88 ALDH1A1 (0.48) ALDH1A1MAOBCYP2D6CYP1A2CYP3A4
SCHEMBL8020337 0.87 MLYCD (0.41) CYP2D6CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL8026762 0.87 ALDH1A1 (0.47) ALDH1A1ALOX5EPORMAOBCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed