SCHEMBL8027615

SCHEMBL8027615

CC1(C)C(=O)N(c2cccc(F)c2)C(=O)N1Cc1ccccc1Cc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.47
TAS2R8 Q9NYW2 9/20 0.46
PGR P06401 1/20 0.42
MCHR1 Q99705 1/20 0.41
IGF1R P08069 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031285 0.91 AR (0.46) ARTAS2R8IGF1R
SCHEMBL8032947 0.90 AR (0.44) ARTAS2R8MCHR1IGF1R
SCHEMBL8030958 0.88 ELANE (0.46) ARTAS2R8IGF1R
SCHEMBL12603161 0.88 AR (0.45) ARTAS2R8PGRMCHR1IGF1R
SCHEMBL8029473 0.88 TAS2R8 (0.46) ARTAS2R8
SCHEMBL1773797 0.88 MGLL (0.45) ARTAS2R8MCHR1IGF1R
SCHEMBL12603148 0.87 AR (0.47) ARTAS2R8IGF1R
SCHEMBL8030817 0.87 AR (0.54) ARTAS2R8IGF1R
SCHEMBL8032989 0.87 AR (0.42) ARTAS2R8MCHR1IGF1R
SCHEMBL8030476 0.86 AR (0.49) ARTAS2R8IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-05-12 US disclosed
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof SANOFI-AVENTIS (FR) 2011-05-12 US disclosed
WO-2009097997-A1 SUBSTITUTED IMIDAZOLIDINE-2,4-DIONES, METHOD FOR THE PRODUCTION THEREOF, MEDICAMENTS CONTAINING SAID COMPOUNDS AND USE THEREOF SANOFI-AVENTIS (FR) 2009-08-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110112097-A1 Substituted imidazoline-2,4-diones, process for preparation thereof, medicaments comprising these compounds and use thereof GIPR, PGC, DDC AR 2449/4885TAS2R8 238/4885PGR 1536/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.