SCHEMBL8028844

SCHEMBL8028844

COc1ccc(C=CC(=O)N(CC(N)C(=O)O)C(=O)C=Cc2ccc(OC)c(OC)c2)cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 1/20 0.58
GRIK2 Q13002 1/20 0.58
APP P05067 4/20 0.57
MAPK1 P28482 2/20 0.57
ALDH1A1 P00352 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
KDM4E B2RXH2 1/20 0.57
HPGD P15428 1/20 0.57
ALOX15 P16050 1/20 0.57
HSD17B10 Q99714 1/20 0.57
NFE2L2 Q16236 1/20 0.56
SNCA P37840 1/20 0.53
KMT2A Q03164 5/20 0.51
MEN1 O00255 3/20 0.51
ABCG2 Q9UNQ0 2/20 0.51
LMNA P02545 1/20 0.50
BCHE P06276 1/20 0.49
MAOA P21397 1/20 0.49
ACHE P22303 1/20 0.49
MAOB P27338 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8030326 0.86 JUN (0.50) GRIK1GRIK2APPALDH1A1SMN1; SMN2
SCHEMBL8028862 0.78 APP (0.57) GRIK1GRIK2APPMAPK1ALDH1A1
SCHEMBL8031856 0.77 JUN (0.51) ALDH1A1SMN1; SMN2KDM4EKMT2AMEN1
SCHEMBL6320958 0.76 APP (0.70) APPMAPK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL6320126 0.76 APP (0.70) APPMAPK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL783249 0.76 APP (0.70) APPMAPK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL10565714 0.74 ALDH1A1 (0.67) APPMAPK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL18699276 0.74 KDM4E (0.67) MAPK1ALDH1A1SMN1; SMN2KDM4EHPGD
SCHEMBL13039641 0.74 NFE2L2 (0.84) APPMAPK1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL29096347 0.74 MAPT (0.61) GRIK1GRIK2APPMAPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000063152-A1 ACETYLATED AND RELATED ANALOGUES OF CHICORIC ACID AS HIV INTEGRASE INHIBITORS THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2000-10-26 WO disclosed