SCHEMBL8029435

SCHEMBL8029435

COC(=O)Cn1ccc2cc(C#N)ccc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.53
NPY5R Q15761 1/20 0.49
ALDH1A1 P00352 6/20 0.48
KDM4E B2RXH2 5/20 0.48
TSHR P16473 4/20 0.48
HSD17B10 Q99714 4/20 0.48
HPGD P15428 3/20 0.48
HTT P42858 2/20 0.48
GLA P06280 1/20 0.48
POLB P06746 2/20 0.47
USP2 O75604 2/20 0.47
PRMT5 O14744 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
FFAR4 Q5NUL3 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RORC P51449 1/20 0.41
MTNR1A P48039 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2470686 0.87 MAPT (0.48) ATMNPY5RALDH1A1KDM4ETSHR
SCHEMBL27844158 0.86 NPY5R (0.45) ATMNPY5RALDH1A1KDM4ETSHR
SCHEMBL3465527 0.83 KMT2A (0.55) NPY5RALDH1A1KDM4ETSHRHSD17B10
SCHEMBL9200019 0.80 MTNR1A (0.60) ATMALDH1A1KDM4EHSD17B10HPGD
SCHEMBL5449877 0.80 ATM (0.57) ATMALDH1A1KDM4EHSD17B10HPGD
SCHEMBL19674140 0.80 ATM (0.57) ATMALDH1A1KDM4EHSD17B10HPGD
SCHEMBL14876504 0.79 NTSR1 (0.57) ATMALDH1A1KDM4EHSD17B10HPGD
SCHEMBL21810428 0.79 NTSR1 (0.57) ATMPRMT5MTNR1AMTNR1BHDAC11
SCHEMBL5637363 0.79 ATM (0.56) ATMALDH1A1KDM4EHSD17B10HPGD
SCHEMBL13699062 0.78 PPARG (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103384661-A Mineralocorticoid receptor antagonists MERCK SHARP & DOHME 2013-11-06 CN claimed
CN-103384661-B Mineralocorticoid receptor antagonists 默沙东公司 2016-08-10 CN disclosed
CN-103384661-A Mineralocorticoid receptor antagonists MERCK SHARP & DOHME 2013-11-06 CN disclosed
US-6043257-A ANTICOAGULANT; PYRIDINE SUBSTITUTED INDAZOLE COMPOUND E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-03-28 US disclosed
US-5886191-A ANTICOAGULANTS DUPONT PHARMACEUTICALS COMPANY (US) 1999-03-23 US disclosed