SCHEMBL8029629

SCHEMBL8029629

Clc1ccc(CN2CCN(CC3CCc4ccccc4O3)CC2)c(Cl)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 4/20 0.67
HTR1A P08908 3/20 0.67
ADRA2A P08913 1/20 0.67
ADRA2B P18089 1/20 0.67
ADRA2C P18825 1/20 0.67
CYP2A13 Q16696 1/20 0.48
HRH3 Q9Y5N1 2/20 0.47
HRH4 Q9H3N8 1/20 0.47
KDM4E B2RXH2 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
ALDH1A1 P00352 1/20 0.47
POLB P06746 1/20 0.47
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
BCHE P06276 1/20 0.45
ACHE P22303 1/20 0.45
BACE1 P56817 1/20 0.45
MAPT P10636 1/20 0.44
CXCR3 P49682 1/20 0.44
SLC6A4 P31645 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029887 0.85 SIGMAR1 (0.83) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8033233 0.81 SIGMAR1 (0.76) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL31061719 0.81 SIGMAR1 (1.00) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8031431 0.81 SIGMAR1 (1.00) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8035733 0.77 HTR1A (0.67) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8035775 0.77 SIGMAR1 (0.81) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8031447 0.77 SIGMAR1 (0.81) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8029628 0.77 SIGMAR1 (0.81) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8035829 0.76 HTR1A (0.65) SIGMAR1HTR1AADRA2AADRA2BADRA2C
SCHEMBL8031437 0.75 ADRA2B (0.60) SIGMAR1HTR1AADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702010-B1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-15 EP disclosed
US-5691340-A CENTRAL NERVOUS SYSTEM DISORDERS, STROKES, CARDIOVASCULAR DISORDERS, ALZHEIMER*S DISEASE OR ANTIINFLAMMATORY AGENTS ADIR ET COMPAGNIE (FR) 1997-11-25 US disclosed
US-5668138-A AFFINITY FOR SIGMA RECEPTORS, CENTRAL NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-09-16 US disclosed
EP-0702010-A1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-03-20 EP disclosed