SCHEMBL8035829

SCHEMBL8035829

COc1ccccc1CN1CCN(CC2CCc3ccccc3O2)CC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.65
SIGMAR1 Q99720 2/20 0.65
ADRA2A P08913 2/20 0.65
ADRA2B P18089 2/20 0.65
ADRA2C P18825 2/20 0.65
GNAI3 P08754 1/20 0.48
CHRM2 P08172 1/20 0.48
CHRM4 P08173 1/20 0.48
CHRM5 P08912 1/20 0.48
CHRM1 P11229 1/20 0.48
CHRM3 P20309 1/20 0.48
DRD2 P14416 2/20 0.47
DRD4 P21917 1/20 0.47
HTR2B P41595 1/20 0.46
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CXCR4 P61073 1/20 0.44
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031437 0.87 ADRA2B (0.60) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8029651 0.82 SIGMAR1 (0.76) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8035733 0.81 HTR1A (0.67) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL31061719 0.79 SIGMAR1 (1.00) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8031431 0.79 SIGMAR1 (1.00) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8029650 0.79 SIGMAR1 (0.71) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL2455767 0.78 ADRA2A (0.57) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8029628 0.78 SIGMAR1 (0.81) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8031447 0.78 SIGMAR1 (0.81) HTR1ASIGMAR1ADRA2AADRA2BADRA2C
SCHEMBL8029629 0.76 SIGMAR1 (0.67) HTR1ASIGMAR1ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1054848-C New benzopyran derivatives, their process of preparation and pharmaceutical compositions which contain them ADIR (FR) 2000-07-26 CN disclosed
EP-0702010-B1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-15 EP disclosed
US-5668138-A AFFINITY FOR SIGMA RECEPTORS, CENTRAL NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-09-16 US disclosed
CN-1132202-A New benzopyran derivatives, their process of preparation and pharmaceutical compositions which contain them ADIR (FR) 1996-10-02 CN disclosed
EP-0702010-A1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-03-20 EP disclosed