SCHEMBL8029940

SCHEMBL8029940

CC(CN1CCN(Cc2ccccc2)CC1)Oc1cccc(F)c1

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
ATM Q13315 1/20 0.52
LTA4H P09960 1/20 0.51
KDM4E B2RXH2 4/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 2/20 0.50
HTT P42858 2/20 0.50
MEN1 O00255 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PPARG P37231 1/20 0.49
PPARA Q07869 1/20 0.49
FAAH O00519 1/20 0.48
HRH3 Q9Y5N1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029920 0.87 LTA4H (0.65) SIGMAR1ATMLTA4HKDM4EKMT2A
SCHEMBL8035768 0.86 SIGMAR1 (0.57) SIGMAR1ATMLTA4HKDM4EALDH1A1
SCHEMBL8033251 0.83 CYP2D6 (0.57) CYP2D6CYP2C9ALOX15TSHRCYP2C19
SCHEMBL8035719 0.79 LTA4H (0.63) SIGMAR1ATMLTA4HKDM4EALDH1A1
SCHEMBL8020078 0.78 LTA4H (0.65) SIGMAR1ATMLTA4HKDM4EKMT2A
SCHEMBL8029621 0.78 LTA4H (0.61) SIGMAR1ATMLTA4HKDM4EALDH1A1
SCHEMBL8035796 0.78 SIGMAR1 (0.68) SIGMAR1LTA4HKDM4EKMT2AALDH1A1
SCHEMBL8029900 0.78 LTA4H (0.57) SIGMAR1ATMLTA4HKMT2AMEN1
SCHEMBL8020087 0.77 MAPK1 (0.60) SIGMAR1CYP2D6CYP2C9TSHRCYP2C19
SCHEMBL16225922 0.76 ALDH1A1 (0.74) SIGMAR1KMT2AALDH1A1MEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702010-B1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-15 EP disclosed
US-5668138-A AFFINITY FOR SIGMA RECEPTORS, CENTRAL NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-09-16 US disclosed
EP-0702010-A1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-03-20 EP disclosed