SCHEMBL8032543

SCHEMBL8032543

CCCc1n[nH]c2c(=O)[nH]c(N(Cc3cccc(N4CCOCC4)c3)CC3CCCCC3)nc12

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 4/20 0.35
HSP90AB1 P08238 3/20 0.35
TTK P33981 1/20 0.34
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
ATM Q13315 6/20 0.33
PIK3C3 Q8NEB9 4/20 0.33
METAP2 P50579 1/20 0.33
PRKDC P78527 1/20 0.33
PARP1 P09874 2/20 0.33
HTR2C P28335 1/20 0.32
PARP14 Q460N5 1/20 0.32
ATR Q13535 1/20 0.32
AGXT P21549 1/20 0.32
TLR7 Q9NYK1 1/20 0.32
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4123059 0.85 PDE5A (0.34) TTKHCRTR1HCRTR2ATMPIK3C3
SCHEMBL4128912 0.85 PDE5A (0.41)
SCHEMBL4142910 0.81 HSP90AA1 (0.37) HSP90AA1HSP90AB1TTKPRKDCAGXT
SCHEMBL4130410 0.79 PARP1 (0.34) ATMPARP1
SCHEMBL4133677 0.78 TPH1 (0.33) HCRTR1HCRTR2ATMPIK3C3METAP2
SCHEMBL4128842 0.78 KDM4E (0.35) HCRTR1HCRTR2ATMPIK3C3PRKDC
SCHEMBL8032549 0.77 PDE5A (0.36) HTR2CTLR7
SCHEMBL8027507 0.75 PDE10A (0.38) ATM
SCHEMBL4136646 0.74 PDE5A (0.43)
SCHEMBL8037857 0.74 PDE5A (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071706-A1 PYRAZOLEPYRIMIDINE COMPOUNDS USEFUL FOR THE TREATMENT OF DEGENERATIVE & INFLAMMATORY DISEASES GALAPAGOS NV (BE) 2009-06-11 WO disclosed