SCHEMBL8033328

SCHEMBL8033328

COC(=O)c1ccc(NCc2cccc(Cl)c2)c(NC(C)=O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.55
HIF1A Q16665 1/20 0.46
MRGPRX4 Q96LA9 1/20 0.46
BRD4 O60885 1/20 0.46
PPM1D O15297 2/20 0.45
MAPT P10636 2/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
ATM Q13315 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
HDAC1 Q13547 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 1/20 0.43
PKM P14618 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
RPS6KB1 P23443 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041888 0.87 ALDH1A1 (0.59) ALDH1A1BRD4MAPTNPC1RAB9A
SCHEMBL4535606 0.85 ALDH1A1 (0.64) ALDH1A1PPM1DMAPTNPC1RAB9A
SCHEMBL8037982 0.83 KDM4E (0.54) ALDH1A1HIF1AMRGPRX4PPM1DMAPT
SCHEMBL8037607 0.80 ALDH1A1 (0.60) ALDH1A1HIF1ABRD4MAPTNPC1
SCHEMBL8024498 0.80 MAPT (0.53) ALDH1A1MAPTNPC1RAB9AMEN1
SCHEMBL22469948 0.78 MRGPRX4 (0.74) HIF1AMRGPRX4PPM1DMAPTNPC1
SCHEMBL31237125 0.76 MRGPRX4 (0.57) ALDH1A1HIF1AMRGPRX4PPM1DMAPT
SCHEMBL15761741 0.75 HIF1A (0.65) ALDH1A1HIF1AMRGPRX4MAPTNPC1
SCHEMBL9402456 0.74 HDAC8 (0.69) ALDH1A1HIF1AMAPTNPC1RAB9A
SCHEMBL8033332 0.74 MEN1 (0.54) ALDH1A1MAPTNPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed