SCHEMBL8033765

SCHEMBL8033765

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NCC2CC2)cc1O

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 3/20 0.43
TDP1 Q9NUW8 1/20 0.40
S1PR1 P21453 5/20 0.39
EPHX2 P34913 2/20 0.38
PDE10A Q9Y233 1/20 0.37
ADRA1D P25100 1/20 0.37
ADRA1A P35348 1/20 0.37
ADRA1B P35368 1/20 0.37
APP P05067 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
HTR4 Q13639 1/20 0.37
PDE4D Q08499 1/20 0.37
MAPK14 Q16539 1/20 0.36
ADRB2 P07550 1/20 0.36
GPR183 P32249 1/20 0.36
APLNR P35414 1/20 0.36
S1PR5 Q9H228 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037415 0.83 S1PR1 (0.41) S1PR1APPADRB2GPR183APLNR
SCHEMBL8040252 0.83 ALDH1A1 (0.41) S1PR1
SCHEMBL8025554 0.82 MTNR1A (0.42) S1PR1APP
SCHEMBL8041411 0.82 S1PR1 (0.43) S1PR1APPTRPV1
SCHEMBL8037435 0.81 PDE10A (0.41) S1PR1PDE10AAPP
SCHEMBL8037394 0.81 POLB (0.46) TDP1S1PR1APP
SCHEMBL8044942 0.81 TDP1 (0.38) CNR2TDP1EPHX2PDE10AADRA1D
SCHEMBL8037440 0.80 PDE10A (0.42) EPHX2PDE10A
SCHEMBL8037831 0.80 ALDH1A1 (0.48)
SCHEMBL8040256 0.80 ALDH1A1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed