SCHEMBL8044942

SCHEMBL8044942

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NCC2CC2)c(C)c1O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
CNR2 P34972 3/20 0.38
EPHX2 P34913 2/20 0.37
PDE4D Q08499 1/20 0.36
MAPK14 Q16539 1/20 0.35
P2RX7 Q99572 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
SLC6A9 P48067 1/20 0.35
PDE10A Q9Y233 1/20 0.34
GAA P10253 1/20 0.34
CNR1 P21554 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033765 0.81 CNR2 (0.43) TDP1CNR2EPHX2PDE4DMAPK14
SCHEMBL8040276 0.78 SMO (0.34) EPHX2PDE4DSLC6A9GAA
SCHEMBL8036155 0.71 MEN1 (0.42) TDP1
SCHEMBL8025559 0.69 MAPT (0.37)
SCHEMBL8035162 0.68 ALDH1A1 (0.41) EPHX2PDE4D
SCHEMBL8037015 0.67 ALDH1A1 (0.45) TDP1
SCHEMBL8034312 0.67 TBXA2R (0.38) EPHX2PDE10A
SCHEMBL8038220 0.67 PPIA (0.42) GAA
SCHEMBL8023142 0.66 ALDH1A1 (0.39)
SCHEMBL8038463 0.66 EPHX2 (0.39) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed