SCHEMBL8033858

SCHEMBL8033858

CCn1nnc(Sc2ncc(NC(=O)c3ccccc3)s2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.49
ALOX15 P16050 2/20 0.45
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
RAB9A P51151 9/20 0.43
NPC1 O15118 8/20 0.43
TP53 P04637 5/20 0.43
SMN1; SMN2 Q16637 6/20 0.42
PKM P14618 1/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
HDAC6 Q9UBN7 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 3/20 0.39
ADORA1 P30542 3/20 0.39
KDR P35968 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8049974 0.92 RAB9A (0.51) ADORA2AALOX15RAB9ANPC1TP53
SCHEMBL8041832 0.90 RAB9A (0.53) ADORA2AALOX15HSD17B10RAB9ANPC1
SCHEMBL1991055 0.90 HDAC6 (0.40) ADORA2AALOX15HPGDRAB9ANPC1
SCHEMBL8047828 0.89 HDAC6 (0.44) ADORA2ARAB9ANPC1SMN1; SMN2HTT
SCHEMBL8047827 0.87 NPC1 (0.41) ADORA2AALOX15RAB9ANPC1TP53
SCHEMBL8033698 0.86 SMN1; SMN2 (0.42) ALOX15HSD17B10RAB9ANPC1TP53
SCHEMBL8050490 0.85 CCNE1 (0.41) ADORA2AALOX15HPGDHSD17B10RAB9A
SCHEMBL8047833 0.84 NPC1 (0.40) ADORA2AALOX15HPGDHSD17B10RAB9A
SCHEMBL8046860 0.83 POLB (0.38) ADORA2AALOX15HPGDHSD17B10RAB9A
SCHEMBL8034295 0.79 NPC1 (0.42) ADORA2ARAB9ANPC1TP53SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed