SCHEMBL8033923

SCHEMBL8033923

Brc1nc(Sc2nnnn2CCc2ccccc2)sc1Br

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
MAPT P10636 2/20 0.37
RAB9A P51151 2/20 0.37
NPC1 O15118 1/20 0.37
UBE2M P61081 3/20 0.37
DCUN1D1 Q96GG9 3/20 0.37
GAA P10253 2/20 0.36
KMT2A Q03164 3/20 0.35
MEN1 O00255 2/20 0.35
SLC6A2 P23975 3/20 0.35
SLC6A4 P31645 3/20 0.35
SLC6A3 Q01959 3/20 0.35
TSHR P16473 3/20 0.35
NPSR1 Q6W5P4 2/20 0.35
KDM4E B2RXH2 2/20 0.35
HTT P42858 2/20 0.35
ATM Q13315 1/20 0.35
LMNA P02545 2/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044545 0.88 ALDH1A1 (0.45) ALDH1A1MAPTRAB9AGAAKMT2A
SCHEMBL8032728 0.85 ALDH1A1 (0.37) ALDH1A1MAPTRAB9ANPC1UBE2M
SCHEMBL8050578 0.81 ALDH1A1 (0.49) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL8050969 0.80 KMT2A (0.39) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL8042957 0.78 HTT (0.41) ALDH1A1MAPTGAAKMT2AMEN1
SCHEMBL8033559 0.77 LMNA (0.47) ALDH1A1MAPTRAB9ANPC1UBE2M
SCHEMBL8042707 0.77 ALDH1A1 (0.46) ALDH1A1MAPTRAB9ANPC1GAA
SCHEMBL8033771 0.77 HSP90AA1 (0.43) ALDH1A1MAPTRAB9ANPC1UBE2M
SCHEMBL8043865 0.76 RAB9A (0.42) ALDH1A1MAPTRAB9ANPC1UBE2M
SCHEMBL8033672 0.76 NPSR1 (0.39) ALDH1A1MAPTRAB9ANPC1UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed