SCHEMBL8034162

SCHEMBL8034162

COc1cc(C(F)(F)F)c(C(=O)N(C)C(=O)NC2CC2)cc1O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.38
APP P05067 1/20 0.38
PDE4B Q07343 1/20 0.37
SMO Q99835 1/20 0.36
GFER P55789 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPT P10636 4/20 0.35
GAA P10253 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 3/20 0.35
KDM4E B2RXH2 2/20 0.35
POLB P06746 1/20 0.35
TAS1R3 Q7RTX0 2/20 0.35
TAS1R1 Q7RTX1 2/20 0.35
TAS1R2 Q8TE23 2/20 0.35
MELK Q14680 1/20 0.35
CCR2 P41597 1/20 0.35
HPGD P15428 2/20 0.34
PTPN7 P35236 2/20 0.34
DUSP3 P51452 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034159 0.95 ALDH1A1 (0.44) GFERALDH1A1MAPTGAAHTT
SCHEMBL8031681 0.83 LRRK2 (0.38) LRRK2APPPDE4BALDH1A1GAA
SCHEMBL8031695 0.82 ALDH1A1 (0.43) GFERALDH1A1MAPTGAAHTT
SCHEMBL8032092 0.82 ALDH1A1 (0.44) GFERALDH1A1MAPTGAAHTT
SCHEMBL8035584 0.81 LRRK2 (0.36) LRRK2APPPDE4BALDH1A1GAA
SCHEMBL8039007 0.81 PTGES (0.41) ALDH1A1MAPTGAAHTTLMNA
SCHEMBL8039269 0.80 ALDH1A1 (0.43) APPALDH1A1LMNAKDM4EHPGD
SCHEMBL8032035 0.80 APP (0.40) APPALDH1A1MAPTGAALMNA
SCHEMBL8035765 0.79 APP (0.38) LRRK2APPALDH1A1MAPTGAA
SCHEMBL8040252 0.79 ALDH1A1 (0.41) LRRK2PDE4BALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed