SCHEMBL8039003

SCHEMBL8039003

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NC2CCC(C)CC2)cc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.47
CNR2 P34972 3/20 0.47
ALDH1A1 P00352 3/20 0.43
TAS1R3 Q7RTX0 2/20 0.43
TAS1R1 Q7RTX1 2/20 0.43
TAS1R2 Q8TE23 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SGMS2 Q8NHU3 1/20 0.42
PPIA P62937 1/20 0.42
GAA P10253 1/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 2/20 0.41
PKM P14618 1/20 0.41
CTSD P07339 1/20 0.41
KDM4E B2RXH2 1/20 0.41
SMPD1 P17405 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025483 0.96 MEN1 (0.46) CNR1CNR2ALDH1A1MEN1KMT2A
SCHEMBL8038995 0.93 ALDH1A1 (0.52) CNR1CNR2ALDH1A1MEN1KMT2A
SCHEMBL8041228 0.92 SGMS2 (0.53) CNR1CNR2ALDH1A1MEN1KMT2A
SCHEMBL8035613 0.82 S1PR1 (0.54) ALDH1A1MEN1KMT2ASGMS2PPIA
SCHEMBL8037213 0.82 MEN1 (0.51) CNR1CNR2ALDH1A1MEN1KMT2A
SCHEMBL8025544 0.82 ALDH1A1 (0.49) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL8039098 0.81 HPGD (0.48) ALDH1A1MEN1KMT2AGAANPC1
SCHEMBL8035618 0.81 APP (0.44) MEN1KMT2ANPC1RAB9APKM
SCHEMBL8025540 0.81 SMN1; SMN2 (0.48) ALDH1A1MEN1KMT2ANPC1RAB9A
SCHEMBL8039269 0.80 ALDH1A1 (0.43) ALDH1A1MEN1KMT2ASGMS2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed