SCHEMBL8041249

SCHEMBL8041249

CN(C(=O)NC1CC1)C(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-]

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
COMT P21964 1/20 0.33
TTR P02766 1/20 0.32
DRD2 P14416 1/20 0.32
SELL P14151 1/20 0.31
SELP P16109 1/20 0.31
SELE P16581 1/20 0.31
NPY5R Q15761 3/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028359 0.88 SMN1; SMN2 (0.35) TAS1R3TAS1R1TAS1R2TTRDRD2
SCHEMBL8035683 0.81 SMYD3 (0.32) TAS1R3TAS1R1TAS1R2COMT
SCHEMBL8035622 0.81 COMT (0.37) COMTALDH1A1
SCHEMBL8041245 0.80 MAPT (0.39) COMTALDH1A1
SCHEMBL8037861 0.79 PPIA (0.41) TAS1R3TAS1R1TAS1R2TTRALDH1A1
SCHEMBL8037250 0.77 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL8025508 0.77 ALDH1A1 (0.37) COMTALDH1A1
SCHEMBL8040243 0.75 PPIA (0.47) ALDH1A1
SCHEMBL8035603 0.75 RAB9A (0.40) ALDH1A1
SCHEMBL8025492 0.74 PPIA (0.49) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed