SCHEMBL8041703

SCHEMBL8041703

CC(C)[C@H](NC(=O)OCc1ccccc1)C(=O)NC(Cc1ccc(OCc2ccccc2)cc1)C(O)C(F)(F)C(=O)NC(c1ccccn1)c1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 5/20 0.49
REN P00797 1/20 0.43
CA2 P00918 1/20 0.42
PSMB11 A5LHX3 5/20 0.42
PSMA7 O14818 5/20 0.42
PSMB1 P20618 5/20 0.42
PSMA1 P25786 5/20 0.42
PSMA2 P25787 5/20 0.42
PSMA3 P25788 5/20 0.42
PSMA4 P25789 5/20 0.42
PSMB8 P28062 5/20 0.42
PSMB9 P28065 5/20 0.42
PSMA5 P28066 5/20 0.42
PSMB4 P28070 5/20 0.42
PSMB6 P28072 5/20 0.42
PSMB5 P28074 5/20 0.42
PSMB10 P40306 5/20 0.42
PSMB3 P49720 5/20 0.42
PSMB2 P49721 5/20 0.42
PSMA6 P60900 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8945683 0.87 CTSD (0.52) CTSDRENPSMB11PSMA7PSMB1
SCHEMBL8054257 0.87 CTSD (0.48) CTSDRENCA2PSMB11PSMA7
SCHEMBL8736745 0.86 CTSD (0.61) CTSDPSMB11PSMA7PSMB1PSMA1
SCHEMBL9095899 0.86 CTSD (0.53) CTSDRENPSMB11PSMA7PSMB1
SCHEMBL7423701 0.86 CTSD (0.51) CTSDRENPSMB11PSMA7PSMB1
SCHEMBL8945567 0.86 CTSD (0.53) CTSDCA2PSMB11PSMA7PSMB1
SCHEMBL8945246 0.86 CTSD (0.53) CTSDRENPSMB11PSMA7PSMB1
SCHEMBL7416869 0.85 MME (0.43) CTSDRENCTSSCTSKITGB3
SCHEMBL7427451 0.85 REN (0.46) RENITGB3ITGA2B
SCHEMBL7419630 0.83 CTSD (0.47) CTSDRENPSMB11PSMA7PSMB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0707564-B1 DIFLUORO STATONE ANALOGS MERRELL PHARMA INC (US) 2000-09-20 EP disclosed
US-6114380-A ANTIVIRAL AGENT; ADMINISTERING TO TREAT HIV INFECTION; N-(4-(N-BENZYLOXYCARBONYL-L-VALYL)AMINO-2,2-DIFLUORO-1,3-DIOXO-5-(4-(2-N -MORPHOLYL)ETHYLOXY)PHENYL-PENTYL)-O-((2-PYRIDYL)METHYL)-D-VALINOL, FOR EXAMPLE MERRELL PHARMACEUTICALS INC. (US) 2000-09-05 US disclosed