SCHEMBL8043075

SCHEMBL8043075

Nc1c(OCc2ccccc2)c(Cl)c2c(c1C(=O)O)CCCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 2/20 0.43
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM3 P20309 1/20 0.40
CLCN2 P51788 1/20 0.40
MCL1 Q07820 1/20 0.40
RXRA P19793 4/20 0.40
RXRB P28702 4/20 0.40
RXRG P48443 3/20 0.40
HPGD P15428 1/20 0.39
HPD P32754 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
MRGPRX4 Q96LA9 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
EGFR P00533 1/20 0.38
ERBB2 P04626 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043037 0.78 PTPN1 (0.44) THRATHRBCHRM4CHRM3CLCN2
SCHEMBL8044819 0.73 TSHR (0.40) DHODHRXRARXRBRXRGHPD
SCHEMBL8043072 0.69 ALDH1A1 (0.35) HPGDKDM4E
SCHEMBL1590791 0.67 ALDH1A1 (0.52) THRATHRBHPGDKDM4ENR4A1
SCHEMBL8884404 0.67 RXRB (0.47) DHODHRXRARXRBRXRGMRGPRX4
SCHEMBL27705561 0.66 MCL1 (0.58) CHRM4CHRM3CLCN2MCL1RXRA
SCHEMBL20659609 0.66 KDM4E (0.46) THRATHRBRXRARXRBHPGD
SCHEMBL8044749 0.66 PIN1 (0.44) RXRARXRBRXRG
SCHEMBL27719021 0.66 THRA (0.44) DHODHTHRATHRBMCL1HPGD
SCHEMBL18702869 0.65 RXRA (0.51) MCL1RXRARXRBRXRGMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686144-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-04-19 EP disclosed
US-5688945-A Compounds ASTRA AKTIEBOLAG (SE) 1997-11-18 US disclosed
US-5661183-A 3-hydroxy anthanilic acid derivatives THE UNIVERSITY OF MARYLAND (US) 1997-08-26 US disclosed
EP-0686144-A1 NEW COMPOUNDS Astra Aktiebolag (SE) 1995-12-13 EP disclosed
WO-1994019315-A1 NEW COMPOUNDS ASTRA AKTIEBOLAG (SE) 1994-09-01 WO disclosed