SCHEMBL8041923

SCHEMBL8041923

O=[N+]([O-])c1ccc2nc(Sc3nnnn3-c3cccc(C(F)(F)F)c3)sc2c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.47
ALDH1A1 P00352 8/20 0.46
MAPT P10636 5/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
HTT P42858 3/20 0.46
LMNA P02545 2/20 0.46
USP2 O75604 1/20 0.46
ALPG P10696 1/20 0.46
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
GAA P10253 1/20 0.43
PKM P14618 1/20 0.43
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
HPGD P15428 2/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
TSHR P16473 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045879 0.87 ALDH1A1 (0.60) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8042814 0.84 PTGS2 (0.40) ALDH1A1MAPTSMN1; SMN2HTTLMNA
SCHEMBL8052209 0.84 ALDH1A1 (0.53) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8049007 0.83 KMT2A (0.45) ALDH1A1MAPTSMN1; SMN2HTTLMNA
SCHEMBL8049105 0.83 PDK1 (0.50) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8033702 0.83 CA2 (0.51) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8042611 0.81 PDK1 (0.53) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8033645 0.80 PDK1 (0.51) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8045309 0.79 ALDH1A1 (0.51) PDK1ALDH1A1MAPTSMN1; SMN2HTT
SCHEMBL8051246 0.79 PDK1 (0.50) PDK1ALDH1A1MAPTSMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed