SCHEMBL8042490

SCHEMBL8042490

C[C@@H](O[Si](C)(C)C(C)(C)C)[C@H]1C(=O)N2C(C(=O)O)=C(Sc3ccccc3C(=O)N3CCCCCC3)[C@H](C)[C@H]12

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ESR1 P03372 1/20 0.34
PTGS1 P23219 1/20 0.34
PDE4A P27815 1/20 0.34
GAA P10253 1/20 0.33
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9834843 0.82 ESR1 (0.37) ESR1PTGS1PDE4A
SCHEMBL8038860 0.82 ESR1 (0.37) ESR1PTGS1PDE4A
SCHEMBL8042493 0.82 SMN1; SMN2 (0.31) HTTALDH1A1SMN1; SMN2GLA
SCHEMBL8834929 0.82 SMN1; SMN2 (0.31) HTTALDH1A1SMN1; SMN2GLA
SCHEMBL9428111 0.77 ELANE (0.36) KMT2AMEN1SMN1; SMN2ESR1PTGS1
SCHEMBL9428941 0.76 CACNA1C (0.36) ESR1PTGS1PDE4A
SCHEMBL9427855 0.76 CACNA1C (0.36) ESR1PTGS1PDE4A
SCHEMBL8046094 0.76 LMNA (0.45) ALDH1A1KMT2AMEN1SMN1; SMN2LMNA
SCHEMBL8039549 0.75 ESR1 (0.33) ALDH1A1ESR1PTGS1PDE4A
SCHEMBL8046007 0.74 CACNA1C (0.36) LMNAESR1PTGS1PDE4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0587436-B1 Process for preparing carbapenem and penem compounds and new compounds involved in that process SANKYO CO (JP) 2000-05-10 EP disclosed
US-5614624-A THIO SUBSTITUTED, ANTIBIOTICS, CHEMICAL INTERMEDIATES SANKYO COMPANY, LIMITED (JP) 1997-03-25 US disclosed
US-5541317-A PENICILLIN DERIVATIVES, CYCLIZATION OF ESTERS OR THIOESTERS SANKYO COMPANY, LIMITED (JP) 1996-07-30 US disclosed