SCHEMBL8043037

SCHEMBL8043037

Cc1c(C)c(C(=O)O)c(N)c(OCc2ccccc2)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MCL1 Q07820 1/20 0.43
POLB P06746 1/20 0.42
GLRA1 P23415 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
MRGPRX4 Q96LA9 3/20 0.41
PTGER1 P34995 1/20 0.40
HPD P32754 1/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
PDE4D Q08499 1/20 0.40
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM3 P20309 1/20 0.40
CLCN2 P51788 1/20 0.40
EDNRA P25101 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13233013 0.79 PTPN1 (0.52) PTPN1POLBGLRA1LMNAHPGD
SCHEMBL22490898 0.78 PDE4D (0.45) PTPN1KDM4EMCL1POLBGLRA1
SCHEMBL8043075 0.78 DHODH (0.43) KDM4EMCL1HPGDMRGPRX4HPD
SCHEMBL31643486 0.74 MAPT (0.49) PTPN1POLBLMNAHPGDPTGER1
SCHEMBL31644450 0.74 ALDH1A1 (0.48) PTPN1KDM4EPOLBLMNAHPGD
SCHEMBL14021700 0.74 MCL1 (0.52) PTPN1KDM4EMCL1GLRA1LMNA
SCHEMBL27739996 0.74 KCNA2 (0.44) PTPN1KDM4EMCL1POLBGLRA1
SCHEMBL27719021 0.74 THRA (0.44) PTPN1MCL1POLBGLRA1LMNA
SCHEMBL31643752 0.73 PTPN1 (0.47) PTPN1POLBGLRA1LMNAHPGD
SCHEMBL26608371 0.73 ALDH1A1 (0.48) PTPN1MCL1POLBGLRA1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686144-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-04-19 EP disclosed
US-5688945-A Compounds ASTRA AKTIEBOLAG (SE) 1997-11-18 US disclosed
US-5661183-A 3-hydroxy anthanilic acid derivatives THE UNIVERSITY OF MARYLAND (US) 1997-08-26 US disclosed
CN-1121344-A New compounds ASTRA AB (SE) 1996-04-24 CN disclosed
EP-0686144-A1 NEW COMPOUNDS Astra Aktiebolag (SE) 1995-12-13 EP disclosed
WO-1994019315-A1 NEW COMPOUNDS ASTRA AKTIEBOLAG (SE) 1994-09-01 WO disclosed