SCHEMBL8043160

SCHEMBL8043160

COc1nsc(N[C@@H](Cc2ccccc2)C(=O)N(C(=O)OCc2ccccc2)[C@@H](C)C(N)=O)n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
ALOX15 P16050 1/20 0.37
ABCB1 P08183 2/20 0.37
CTSL P07711 4/20 0.36
CTSB P07858 2/20 0.36
CTSS P25774 2/20 0.36
CTSK P43235 2/20 0.36
POLB P06746 1/20 0.35
CAPN1 P07384 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
THRB P10828 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450371 0.81 XIAP (0.39) ALDH1A1ALOX15ABCB1MEN1KMT2A
SCHEMBL7640967 0.79 ATM (0.47) ALDH1A1ALOX15POLBTHRBCYP2C9
SCHEMBL7409774 0.72 CTSL (0.54) ALDH1A1ALOX15CTSLCTSBCTSS
SCHEMBL30297616 0.72 ALDH1A1 (0.51) ALDH1A1ABCB1KMT2A
SCHEMBL7450374 0.71 CTSL (0.50) ALDH1A1ALOX15CTSLCTSBCTSS
SCHEMBL7409777 0.71 SLC15A1 (0.41) ALDH1A1ALOX15ABCB1CTSLCTSB
SCHEMBL7637777 0.70 ELANE (0.42)
SCHEMBL27899925 0.67 ABCB1 (0.44) ALDH1A1ABCB1CTSLCTSBCTSS
SCHEMBL7994098 0.66 ALDH1A1 (0.50) ALDH1A1ALOX15ABCB1CTSLCTSB
SCHEMBL11341463 0.65 CTSK (0.47) CTSLCTSBCTSSCTSKCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114537-A 1,2,4-THIADIAZOLE COMPOUND IS USEFUL FOR TRAPPING THIOL COMPOUNDS AND SELECTIVELY CHANGING THIOLS TO DISULFIDE COMPOUNDS APOTEX INC. (CA) 2000-09-05 US disclosed