SCHEMBL8043428

SCHEMBL8043428

Cc1nc(Sc2nccs2)n[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 1/20 0.43
FBP1 P09467 4/20 0.42
PDK1 Q15118 1/20 0.42
RAB9A P51151 4/20 0.37
HTR7 P34969 1/20 0.37
POLB P06746 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 2/20 0.34
LMNA P02545 2/20 0.34
TSHR P16473 2/20 0.34
HTT P42858 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
FLT3 P36888 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048057 0.76 RAB9A (0.39) EGLN1RAB9APOLBSMN1; SMN2LMNA
SCHEMBL8043319 0.73 KDM4E (0.53) FBP1PDK1RAB9APOLBSMN1; SMN2
SCHEMBL8043572 0.71 EGLN1 (0.38) EGLN1RAB9APOLBSMN1; SMN2NPC1
SCHEMBL7114230 0.71 FBP1 (0.70) FBP1PDK1HTR7TSHRFLT3
SCHEMBL8033034 0.70 FBP1 (0.47) FBP1PDK1HTR7SMN1; SMN2FLT3
SCHEMBL8050307 0.68 HTR1A (0.47) EGLN1RAB9AHTR7SMN1; SMN2NPC1
SCHEMBL8043078 0.67 FBP1 (0.47) FBP1PDK1RAB9AHTR7NPC1
SCHEMBL8048521 0.67 POLB (0.36) EGLN1RAB9APOLBSMN1; SMN2LMNA
SCHEMBL8045613 0.66 RAB9A (0.44) RAB9APOLBSMN1; SMN2NPC1LMNA
SCHEMBL17274031 0.66 FBP1 (0.45) FBP1PDK1HTR7FLT3KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed