SCHEMBL8044729

SCHEMBL8044729

Fc1ccc(-c2nnc(S)s2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
CSNK2A2 P19784 1/20 0.43
CSNK2A1 P68400 1/20 0.43
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
KDM4E B2RXH2 2/20 0.41
HDAC1 Q13547 2/20 0.40
HRH3 Q9Y5N1 1/20 0.40
HDAC2 Q92769 1/20 0.40
PSMD14 O00487 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
BLM P54132 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14557099 0.89 KDM4E (0.43) SMN1; SMN2CSNK2A2CSNK2A1RAB9ANPC1
SCHEMBL8047389 0.79 CA1 (0.49) SMN1; SMN2RAB9ANPC1KDM4EHDAC1
SCHEMBL8050989 0.79 ALDH1A1 (0.60) SMN1; SMN2KMT2AMEN1RAB9ANPC1
SCHEMBL9360268 0.79 GAA (0.60) SMN1; SMN2KMT2AMEN1RAB9ANPC1
SCHEMBL972899 0.79 MGAM (0.60) SMN1; SMN2KMT2AMEN1RAB9ANPC1
SCHEMBL8050331 0.79 KIF11 (0.44) SMN1; SMN2KMT2AMEN1RAB9ANPC1
SCHEMBL969040 0.78 ALDH1A1 (0.52) SMN1; SMN2KMT2AMEN1RAB9ANPC1
SCHEMBL8047555 0.77 KDM4E (0.65) SMN1; SMN2KMT2AMEN1RAB9ANPC1
SCHEMBL3826842 0.77 HDAC1 (0.44) SMN1; SMN2KMT2AMEN1CSNK2A2CSNK2A1
SCHEMBL969939 0.77 KDM4E (0.59) SMN1; SMN2KMT2AMEN1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112244031-A Application of thiothiadiazole-containing nitrothiazole compound in prevention and treatment of agricultural plant diseases 兰州大学 2021-01-22 CN disclosed
CN-104292224-B Containing replacing 1,3,4-thiophene () diazole thioether benzothiazole amide derivatives and its preparation method and application 贵州大学 2016-07-06 CN disclosed
CN-104292224-A Benzothiazole amide derivatives containing substituted 1,3,4-thiadiazole (oxadiazole) thioether as well as preparation method and application of derivatives UNIV GUIZHOU 2015-01-21 CN disclosed
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed