SCHEMBL8044770

SCHEMBL8044770

FC(F)(F)c1nnc(Sc2nccs2)s1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 12/20 0.43
PDK1 Q15118 1/20 0.42
ALDH1A1 P00352 1/20 0.36
HTR7 P34969 1/20 0.33
FDPS P14324 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33
GABRA5 P31644 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRA2 P47869 1/20 0.33
HTT P42858 1/20 0.32
FLT3 P36888 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7114230 0.75 FBP1 (0.70) FBP1PDK1ALDH1A1HTR7FDPS
SCHEMBL8048536 0.74 FBP1 (0.47) FBP1PDK1ALDH1A1HTR7
SCHEMBL8043078 0.74 FBP1 (0.47) FBP1PDK1ALDH1A1HTR7GABRA1
SCHEMBL8045097 0.72 RAB9A (0.35) ALDH1A1HTTNPC1RAB9A
SCHEMBL8043975 0.72 ALDH1A1 (0.35) ALDH1A1
SCHEMBL8046775 0.70 FBP1 (0.42) FBP1PDK1ALDH1A1HTR7FDPS
SCHEMBL8047678 0.70 FBP1 (0.42) FBP1PDK1ALDH1A1HTR7FDPS
SCHEMBL8048705 0.70 FBP1 (0.46) FBP1PDK1ALDH1A1HTR7FDPS
SCHEMBL13814464 0.69 ALDH1A1 (0.50) FBP1ALDH1A1HTTNPC1RAB9A
SCHEMBL8045096 0.68 PDPK1 (0.51) FBP1PDK1ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed