SCHEMBL8044910

SCHEMBL8044910

Cc1ccc(-n2nnnc2Sc2nc3ccc(S(C)(=O)=O)cc3s2)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.43
RAB9A P51151 6/20 0.43
SMN1; SMN2 Q16637 5/20 0.43
ALDH1A1 P00352 5/20 0.43
TP53 P04637 4/20 0.43
KDM4E B2RXH2 2/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
PKM P14618 1/20 0.41
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 2/20 0.40
HPGD P15428 1/20 0.40
ILK Q13418 1/20 0.38
POLB P06746 3/20 0.37
ACP1 P24666 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047942 0.89 PKM (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8033619 0.87 PKM (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8050340 0.87 KMT2A (0.46) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8044412 0.85 SMN1; SMN2 (0.44) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8052304 0.84 ALDH1A1 (0.49) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8050208 0.83 PDK1 (0.52) NPC1RAB9ASMN1; SMN2ALDH1A1TSHR
SCHEMBL8047829 0.82 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8033160 0.82 PKM (0.51) SMN1; SMN2ALDH1A1TP53TSHRPKM
SCHEMBL8048328 0.82 PKM (0.41) NPC1RAB9ASMN1; SMN2ALDH1A1TP53
SCHEMBL8033856 0.82 PKM (0.46) NPC1RAB9ASMN1; SMN2ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed