SCHEMBL8045430

SCHEMBL8045430

CS(=O)(=O)O.CS(=O)(=O)O.Cc1cc(C)c2cccc(OCc3c(Cl)ccc(S(=O)(=O)N4CCC[C@H]4C(=O)NCCCNC(=O)c4ccc(C=NN)cc4)c3Cl)c2n1

nearest known ligand 0.82

Known targets — ChEMBL curated mechanism

ABL1ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB2AGTR1BCL2BCL2A1BCL2L1BCL2L10BCL2L2BCRBRAFCHRM1CHRNA10CHRNA9DRD1DRD2DRD3DRD4DRD5EGFRF2FLT1FLT4GCKGHSRGNRHRGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHTR1AHTR1BHTR1DHTR2AHTR2CHTR3AIDH2KDRKITMAOBMCL1MTTPPP4HBPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PIKFYVEROCK1ROCK2SLC18A2SLC6A2SLC6A3SLC6A4TACR1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8gyrAgyrBparCparEpol

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 4/20 0.82
RORC P51449 16/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6948878 0.99 BDKRB2 (0.82) BDKRB2RORC
SCHEMBL6945418 0.99 BDKRB2 (0.84) BDKRB2RORC
Hydrochloric Acid SCHEMBL8045266 0.98 BDKRB2 (0.83) BDKRB2RORC
SCHEMBL6950086 0.98 BDKRB2 (0.81) BDKRB2RORC
Hydrochloric Acid SCHEMBL8040364 0.98 BDKRB2 (0.80) BDKRB2RORC
SCHEMBL6953309 0.96 BDKRB2 (0.80) BDKRB2RORC
Hydrochloric Acid SCHEMBL8041915 0.96 BDKRB2 (0.79) BDKRB2RORC
SCHEMBL8042006 0.94 BDKRB2 (0.74) BDKRB2RORC
SCHEMBL6947379 0.94 BDKRB2 (0.79) BDKRB2RORC
SCHEMBL8028477 0.93 BDKRB2 (0.72) BDKRB2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6063791-A N-benzenesulfonyl-L-proline derivatives, method for preparing and therapeutic use FOURNIER INDUSTRIE ET SANTE (FR) 2000-05-16 US disclosed