SCHEMBL8046744

SCHEMBL8046744

c1ccc2sc(Sc3nnnn3-c3nccs3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
HPGD P15428 5/20 0.48
L3MBTL1 Q9Y468 3/20 0.48
TSHR P16473 2/20 0.48
SMN1; SMN2 Q16637 5/20 0.45
MAPT P10636 4/20 0.45
HTT P42858 3/20 0.45
KDM4E B2RXH2 1/20 0.45
HSD17B10 Q99714 2/20 0.41
ADRA2A P08913 1/20 0.41
FBP1 P09467 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
DRD2 P14416 1/20 0.41
ALOX15 P16050 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
DRD1 P21728 1/20 0.41
MC5R P33032 1/20 0.41
OPRM1 P35372 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047505 0.82 HSP90AA1 (0.41) ALDH1A1HPGDL3MBTL1TSHRSMN1; SMN2
SCHEMBL8042637 0.81 HPGD (0.41) ALDH1A1HPGDL3MBTL1TSHRSMN1; SMN2
SCHEMBL8043423 0.81 ALDH1A1 (0.50) ALDH1A1HPGDL3MBTL1TSHRSMN1; SMN2
SCHEMBL8046990 0.81 ALDH1A1 (0.47) ALDH1A1HPGDL3MBTL1TSHRSMN1; SMN2
SCHEMBL8042782 0.80 PKM (0.39) ALDH1A1HPGDSMN1; SMN2MAPTHTT
SCHEMBL8044167 0.80 PDK1 (0.51) ALDH1A1HPGDTSHRSMN1; SMN2MAPT
SCHEMBL8046562 0.80 ALDH1A1 (0.70) ALDH1A1HPGDL3MBTL1TSHRSMN1; SMN2
SCHEMBL8043970 0.79 KMT2A (0.43) ALDH1A1TSHRSMN1; SMN2MAPTHTT
SCHEMBL8045872 0.78 FBP1 (0.40) ALDH1A1HPGDSMN1; SMN2MAPTHTT
SCHEMBL8044672 0.77 TP53 (0.32) ALDH1A1SMN1; SMN2MAPTHTTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed