SCHEMBL8049892

SCHEMBL8049892

CCOC(=O)CCCCCCC(C#N)(c1ccccc1)c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.48
KCNA3 P22001 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.46
CYP4F2 P78329 1/20 0.46
CYP4A11 Q02928 1/20 0.46
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
CYP2D6 P10635 1/20 0.44
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
NAMPT P43490 1/20 0.42
ALOX5 P09917 1/20 0.41
CCR1 P32246 1/20 0.41
FAAH O00519 2/20 0.41
TOP2A P11388 1/20 0.41
TBXAS1 P24557 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044856 1.00 OPRM1 (0.48) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL8046235 0.99 OPRM1 (0.49) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL7830375 0.95 OPRM1 (0.50) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL8047298 0.93 OPRM1 (0.44) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL8046383 0.90 CYP4F2 (0.40) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL7826967 0.89 KCNA3 (0.52) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL8035567 0.88 CA12 (0.40) OPRM1KCNA3CYP4F2CYP4A11ALDH1A1
SCHEMBL8035702 0.88 SMN1; SMN2 (0.40) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL8047345 0.88 KCNA3 (0.40) OPRM1KCNA3SMN1; SMN2CYP4F2CYP4A11
SCHEMBL8053206 0.87 FAAH (0.44) OPRM1KCNA3CYP4F2CYP4A11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0749957-B1 Aromatic hydroxamic acid compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-04-26 EP disclosed
US-5891916-A ANTINEUROGEGERATIVE AGENT TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-04-06 US disclosed
EP-0749957-A1 Aromatic hydroxamic acid compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1996-12-27 EP disclosed