SCHEMBL8050815

SCHEMBL8050815

Clc1ccc(NC2COc3ccccc32)nn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.46
ALDH1A1 P00352 3/20 0.41
GAA P10253 3/20 0.39
MAPT P10636 2/20 0.39
HTR1A P08908 1/20 0.37
HTR1D P28221 1/20 0.37
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
RIPK1 Q13546 1/20 0.35
CYP2D6 P10635 2/20 0.34
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
DRD2 P14416 1/20 0.33
DRD3 P35462 1/20 0.33
MAPK1 P28482 1/20 0.33
GLS O94925 1/20 0.33
LTB4R Q15722 1/20 0.33
LTB4R2 Q9NPC1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8054302 0.86 LRRK2 (0.41) P2RX7ALDH1A1GAAMAPTHTR1A
SCHEMBL8060412 0.86 LRRK2 (0.41) P2RX7ALDH1A1GAAMAPTHTR1A
SCHEMBL3829666 0.71 P2RX7 (0.45) P2RX7DRD2DRD3MAPK1LTB4R
SCHEMBL3409292 0.68 PLAU (0.39) P2RX7ALDH1A1GAAMAPTHTR1A
SCHEMBL3404302 0.68 BACE1 (0.37) P2RX7ALDH1A1MAPTHTR1AKDM4E
SCHEMBL6369306 0.67 ADRA2A (0.58) P2RX7HTR1ACYP2D6LTB4RLTB4R2
SCHEMBL22655135 0.67 GAA (0.52) ALDH1A1GAAMAPTKDM4ELMNA
SCHEMBL29565663 0.67 GAA (0.52) ALDH1A1GAAMAPTKDM4ELMNA
SCHEMBL24915634 0.67 LTB4R (0.45) P2RX7CYP2D6SLC6A2SLC6A4DRD2
SCHEMBL506553 0.67 PDPK1 (0.46) CYP2D6SLC6A2SLC6A4LTB4RLTB4R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009050227-A1 PYRIDAZINE DERIVATIVES FOR INHIBITING BETA AMYLOID PEPTIDE PRODUCTION GLAXO GROUP LIMITED (GB) 2009-04-23 WO disclosed