SCHEMBL8052849

SCHEMBL8052849

NC1CCCN1C1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
THRB P10828 1/20 0.30
MEN1 O00255 1/20 0.30
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL962787 0.95 HTR6 (0.31) KMT2ATHRBMEN1DPP4
SCHEMBL7870406 0.95 HTR6 (0.31) KMT2ATHRBMEN1DPP4
SCHEMBL729174 0.95 HTR6 (0.31) KMT2ATHRBMEN1DPP4
SCHEMBL8146446 0.72 HTR6 (0.47)
SCHEMBL11735212 0.70 ALDH1A1 (0.33) ALDH1A1SMN1; SMN2KMT2ACYP3A4CYP2C9
SCHEMBL5872327 0.70 HRH3 (0.38) ALDH1A1SMN1; SMN2KMT2ACYP3A4CYP2C9
SCHEMBL10721919 0.70 EPHX1 (0.33) ALDH1A1SMN1; SMN2KMT2ACYP3A4CYP2C9
SCHEMBL3246436 0.70 EPHX1 (0.33) ALDH1A1SMN1; SMN2KMT2ACYP3A4CYP2C9
SCHEMBL10721961 0.70 EPHX1 (0.33) ALDH1A1SMN1; SMN2KMT2ACYP3A4CYP2C9
SCHEMBL7019251 0.70 EPHX1 (0.33) ALDH1A1SMN1; SMN2KMT2ACYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080760-A TREATING BENIGN PROSTATIC HYPERPLASIA; COMPLEMENT SLOWER-ACTING THERAPEUTICS BY PROVIDING ACUTE RELIEF; INDUCE RELAXATION OF THE LOWER URINARY TRACT TO DECREASE DIFFICULTY IN URINATION AND SEXUAL DYSFUNCTION MERCK & CO., INC. (US) 2000-06-27 US disclosed
EP-1003511-A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2000-05-31 EP disclosed
WO-1998057639-A1 ALPHA 1aADRENERGIC RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1998-12-23 WO disclosed
US-4041032-A ANTIEMATICS, GASTRIC MOTILITY STIMULANTS YAMANOUCHI PHARMACEUTICAL CO., LTD. (JA) 1977-08-09 US disclosed