SCHEMBL8071844

SCHEMBL8071844

Cc1nc(N)cc(C(=O)NCc2cccc(OCCO)c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 8/20 0.49
ROCK2 O75116 6/20 0.49
CYP3A4 P08684 4/20 0.49
CYP2D6 P10635 4/20 0.49
CYP2C9 P11712 4/20 0.49
ADORA3 P0DMS8 2/20 0.47
ADORA2A P29274 2/20 0.47
ADORA2B P29275 2/20 0.47
ADORA1 P30542 2/20 0.47
MMP13 P45452 5/20 0.46
KDM4E B2RXH2 2/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
CHRM4 P08173 1/20 0.43
PRKACA P17612 2/20 0.43
PRKX P51817 2/20 0.43
PRKCQ Q04759 2/20 0.43
GRK5 P34947 1/20 0.43
GSK3A P49840 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8055078 0.81 MMP13 (0.47) ROCK1ROCK2MMP13ALDH1A1
SCHEMBL8058261 0.80 MMP13 (0.51) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8055231 0.76 MMP13 (0.58) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL3685174 0.73 MMP13 (0.60) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8067349 0.72 MMP13 (0.55) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL24674846 0.71 ROCK2 (0.47) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL13837856 0.70 MMP13 (0.53) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL8070937 0.70 MMP13 (0.57) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL1240006 0.70 ALDH1A1 (0.48) ROCK1ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL31567851 0.70 TSHR (0.62) MMP13ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009016498-A1 PYRIMIDINE AND PYRIDINE DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS PFIZER INC. (US) 2009-02-05 WO disclosed