SCHEMBL8066489

SCHEMBL8066489

COc1ccc(S(=O)(=O)N2CCCC2CNC(=O)NC23CC4C[C@@H]5CC(C2)C3(C4)C5)c(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.43
NPC1 O15118 1/20 0.43
PAX8 Q06710 1/20 0.41
FKBP1A P62942 1/20 0.38
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060003 0.98 RAB9A (0.41) RAB9ANPC1PAX8FKBP1ATSHR
SCHEMBL8062528 0.86 RAB9A (0.50) RAB9ANPC1PAX8
SCHEMBL4538117 0.85 FKBP1A (0.48) RAB9ANPC1PAX8FKBP1A
SCHEMBL8068365 0.84 RAB9A (0.42) RAB9ANPC1PAX8FKBP1ATSHR
SCHEMBL8062049 0.82 CYP19A1 (0.40) FKBP1ATSHR
SCHEMBL4542922 0.82 RAB9A (0.49) RAB9ANPC1PAX8HCRTR1HCRTR2
SCHEMBL8062526 0.80 NPC1 (0.38) RAB9ANPC1
SCHEMBL4537168 0.80 RAB9A (0.47) RAB9ANPC1PAX8FKBP1ATSHR
SCHEMBL8062873 0.79 HCRTR1 (0.42) HCRTR1
SCHEMBL8066636 0.79 RAB9A (0.46) RAB9APAX8TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed