SCHEMBL8066788

SCHEMBL8066788

O=c1[nH]c2cc(C=Cc3cccnc3)ccc2c(=O)c2[nH]nnc12

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PADI4 Q9UM07 8/20 0.40
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
TDO2 P48775 3/20 0.38
IDO1 P14902 1/20 0.38
MEN1 O00255 1/20 0.37
MAPT P10636 1/20 0.37
KMT2A Q03164 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
TTK P33981 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8068010 0.92 PADI4 (0.43) PADI4NPC1RAB9ATDO2IDO1
SCHEMBL8073308 0.86 IP6K1 (0.41) NPC1RAB9AMAPTALDH1A1TTK
SCHEMBL8073292 0.86 IP6K1 (0.41) NPC1RAB9AMAPTALDH1A1TTK
SCHEMBL8069062 0.83 IP6K1 (0.46) PADI4NPC1RAB9AMEN1MAPT
SCHEMBL8069058 0.83 IP6K1 (0.46) PADI4NPC1RAB9AMEN1MAPT
SCHEMBL7825535 0.80 KIF11 (0.43) TTK
SCHEMBL8058054 0.80 ALDH1A1 (0.41) NPC1RAB9AMEN1MAPTKMT2A
SCHEMBL8058059 0.80 ALDH1A1 (0.41) NPC1RAB9AMEN1MAPTKMT2A
SCHEMBL7825711 0.79 CCNB2 (0.37)
SCHEMBL7825041 0.79 CCNB2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2000239260-A PRODUCTION OF OPTICALLY ACTIVE 2-PIPERAZINECARBOXYLIC ACID KOEI CHEM CO LTD 2000-09-05 JP disclosed
US-6093714-A AN ANTIALLERGENS FOR TREATMENT AND PREVENTION OF BRONCHIAL ASTHMA, ECZEMA, HIVES, ALLERGIC GASTROINTESTINAL TROUBLES, ALLERGIC RHINITIS, ALLERGIC CONJUNCTIVITIS MEIJI SEIKA KAISHA, LTD. (JP) 2000-07-25 US disclosed