SCHEMBL8068409

SCHEMBL8068409

CCOC(=O)c1[nH]c2cccc3c2c1CCC3=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
GAA P10253 2/20 0.48
MAP3K5 Q99683 1/20 0.47
PARP1 P09874 3/20 0.46
AURKA O14965 1/20 0.46
MAPK10 P53779 1/20 0.46
RIPK1 Q13546 1/20 0.46
BRD4 O60885 1/20 0.45
MAPT P10636 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KDM4E B2RXH2 5/20 0.43
HTR6 P50406 2/20 0.43
HSD17B10 Q99714 2/20 0.42
TUBB4A P04350 2/20 0.42
TUBB P07437 2/20 0.42
TUBA3C P0DPH7 2/20 0.42
TUBA1B P68363 2/20 0.42
TUBA4A P68366 2/20 0.42
TUBB4B P68371 2/20 0.42
TUBB3 Q13509 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068336 0.79 BRD4 (0.49) ALDH1A1AURKAMAPK10RIPK1BRD4
SCHEMBL8074787 0.76 MTNR1A (0.45) ALDH1A1MAP3K5AURKAMAPK10RIPK1
SCHEMBL11630902 0.76 ALDH1A1 (0.60) ALDH1A1GAAMAPK10MAPTKDM4E
SCHEMBL8059219 0.74 KDM4E (0.44) ALDH1A1GAAAURKAMAPK10RIPK1
SCHEMBL5002514 0.72 PARP1 (0.59) PARP1
SCHEMBL24074529 0.72 KDM4E (0.48) ALDH1A1MAP3K5MAPTKDM4EHTR6
SCHEMBL7566334 0.72 MAPT (0.53) ALDH1A1MAP3K5MAPTKDM4EHTR6
SCHEMBL8070000 0.72 PARP1 (0.50) ALDH1A1GAAPARP1MAPTKDM4E
SCHEMBL24073034 0.72 NPC1 (0.48) ALDH1A1GAAMAP3K5MAPTNPSR1
SCHEMBL8070221 0.72 MEN1 (0.48) ALDH1A1GAAMAPTKDM4EHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0803501-B1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMA (JP) 2000-07-05 EP disclosed
EP-0803501-A1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-29 EP disclosed