SCHEMBL8074787

SCHEMBL8074787

CCOC(=O)c1[nH]c2cccc3c2c1CCC3O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 2/20 0.45
MTNR1B P49286 2/20 0.45
KDM4E B2RXH2 8/20 0.43
AURKA O14965 1/20 0.42
MAPK10 P53779 1/20 0.42
RIPK1 Q13546 1/20 0.42
HTR6 P50406 2/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 3/20 0.41
TUBB4A P04350 2/20 0.40
TUBB P07437 2/20 0.40
TUBA3C P0DPH7 2/20 0.40
TUBA1B P68363 2/20 0.40
TUBA4A P68366 2/20 0.40
TUBB4B P68371 2/20 0.40
TUBB3 Q13509 2/20 0.40
TUBB2A Q13885 2/20 0.40
TUBB8 Q3ZCM7 2/20 0.40
TUBA3E Q6PEY2 2/20 0.40
TUBA1A Q71U36 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059219 0.93 KDM4E (0.44) MTNR1AMTNR1BKDM4EAURKAMAPK10
SCHEMBL8068336 0.77 BRD4 (0.49) KDM4EAURKAMAPK10RIPK1HTR6
SCHEMBL8068409 0.76 ALDH1A1 (0.48) KDM4EAURKAMAPK10RIPK1HTR6
SCHEMBL9364035 0.75 HSD11B1 (0.42) MTNR1AMTNR1BKDM4EHTR6ALDH1A1
SCHEMBL8070427 0.71 PARP1 (0.38) KDM4EALDH1A1HSD17B10HPGDHTR1A
SCHEMBL8070432 0.70 PARP1 (0.37) KDM4EALDH1A1HTR1ADRD2
SCHEMBL6624045 0.70 PARP1 (0.48) DRD2
SCHEMBL27408415 0.70 ALDH1A1 (0.54) KDM4EHTR6ALDH1A1HSD17B10TUBB4A
SCHEMBL21485065 0.69 DRD2 (0.45) MAPK10ALDH1A1HSD17B10TSHRDRD2
SCHEMBL8069946 0.69 KMT2A (0.41) KDM4EALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0803501-B1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMA (JP) 2000-07-05 EP disclosed
EP-0803501-A1 Substituted guanidine derivatives and their use as Na+/H+ exchange inhibitors SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-29 EP disclosed