SCHEMBL8074157

SCHEMBL8074157

C=CCOC(=O)c1nc2ccccc2c(O)c1C(=O)OCC=C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
GABRA1 P14867 1/20 0.43
GABRB1 P18505 1/20 0.43
GABRG2 P18507 1/20 0.43
GABRB3 P28472 1/20 0.43
GABRA5 P31644 1/20 0.43
GABRA3 P34903 1/20 0.43
GABRA2 P47869 1/20 0.43
GABRB2 P47870 1/20 0.43
GABRA4 P48169 1/20 0.43
GABRE P78334 1/20 0.43
GABRA6 Q16445 1/20 0.43
GABRG1 Q8N1C3 1/20 0.43
GABRG3 Q99928 1/20 0.43
GABRQ Q9UN88 1/20 0.43
MEN1 O00255 5/20 0.43
KMT2A Q03164 5/20 0.43
ALDH1A1 P00352 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528103 0.81 CYP3A4 (0.50) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL8546392 0.77 ADORA3 (0.53) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL11775934 0.75 CYP3A4 (0.53) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL11799224 0.75 CYP3A4 (0.65) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL8569494 0.75 MEN1 (0.56) MEN1KMT2AALDH1A1POLBTSHR
SCHEMBL28797295 0.74 KDM4E (0.53) MEN1KMT2AALDH1A1LMNASMN1; SMN2
SCHEMBL28662473 0.73 CYP3A4 (0.57) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL7071011 0.72 CYP3A4 (0.53) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL11090058 0.72 KDM4E (0.49) CYP3A4GABRPGABRDGABRA1GABRB1
SCHEMBL8539340 0.71 ALDH1A1 (0.52) CYP3A4GABRPGABRDGABRA1GABRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6103721-A TREATMENT OF STROKE ANOXIA; ANTIHYPERGLYCEMIC,-ISCHEMIC AND -EPILEPTIC AGENTS ZENECA LIMITED (GB) 2000-08-15 US disclosed