SCHEMBL9528103

SCHEMBL9528103

C=CCOC(=O)c1nnc2ccccc2c1O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.50
ALDH1A1 P00352 4/20 0.44
HSD17B10 Q99714 2/20 0.44
TSHR P16473 1/20 0.44
RHOA P61586 1/20 0.42
LCK P06239 1/20 0.40
MAP2K3 P46734 1/20 0.40
MAP2K6 P52564 1/20 0.40
BTK Q06187 1/20 0.40
MAP3K19 Q56UN5 1/20 0.40
NEK10 Q6ZWH5 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
SNCA P37840 1/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10861354 0.81 KDM4E (0.51) ALDH1A1TSHRKDM4EMEN1KMT2A
SCHEMBL8074157 0.81 CYP3A4 (0.48) CYP3A4ALDH1A1HSD17B10TSHRRHOA
SCHEMBL1123696 0.76 KDM4E (0.47) ALDH1A1TSHRLCKMAP2K3MAP2K6
SCHEMBL8546392 0.74 ADORA3 (0.53) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL7706331 0.72 LCK (0.51) ALDH1A1HSD17B10TSHRLCKMAP2K3
SCHEMBL31371878 0.72 LCK (0.51) ALDH1A1HSD17B10TSHRLCKMAP2K3
SCHEMBL11775934 0.71 CYP3A4 (0.53) CYP3A4ALDH1A1HSD17B10TSHRRHOA
SCHEMBL9525498 0.71 LCK (0.50) ALDH1A1LCKMAP2K3MAP2K6BTK
SCHEMBL11799224 0.71 CYP3A4 (0.65) CYP3A4ALDH1A1HSD17B10TSHRRHOA
SCHEMBL6890781 0.71 LCK (0.69) ALDH1A1LCKMAP2K3MAP2K6BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0277791-B1 CINNOLINE-CARBOXAMIDES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.r.l. (IT) 1993-06-02 EP disclosed
US-4826837-A IMMUNOMODULATORS FARMITALIA CARLO ERBA S.R.L. (IT) 1989-05-02 US disclosed
EP-0277791-A2 Cinnoline-carboxamides and process for their preparation FARMITALIA CARLO ERBA S.r.l. (IT) 1988-08-10 EP disclosed