SCHEMBL8546392

SCHEMBL8546392

C=CCOC(=O)c1nc(N)nc2ccccc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.53
ALDH1A1 P00352 2/20 0.50
HSD17B10 Q99714 2/20 0.50
TSHR P16473 1/20 0.50
CYP3A4 P08684 1/20 0.49
HSP90AA1 P07900 2/20 0.47
HSP90AB1 P08238 2/20 0.47
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRB1 P18505 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44
GABRA4 P48169 1/20 0.44
GABRE P78334 1/20 0.44
GABRA6 Q16445 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27890879 0.81 KMT2A (0.53) ADORA3ALDH1A1HSP90AA1HSP90AB1ADORA2A
SCHEMBL8539340 0.77 ALDH1A1 (0.52) ALDH1A1HSD17B10TSHRCYP3A4GABRP
SCHEMBL8074157 0.77 CYP3A4 (0.48) ALDH1A1HSD17B10TSHRCYP3A4GABRP
SCHEMBL28293697 0.77 ADORA3 (0.61) ADORA3ALDH1A1HSD17B10TSHRHSP90AA1
SCHEMBL11775934 0.76 CYP3A4 (0.53) ALDH1A1HSD17B10TSHRCYP3A4HSP90AA1
SCHEMBL3088381 0.74 ADORA3 (0.66) ADORA3ALDH1A1HSD17B10HSP90AA1HSP90AB1
SCHEMBL9528103 0.74 CYP3A4 (0.50) ALDH1A1HSD17B10TSHRCYP3A4GABRP
SCHEMBL28288558 0.73 CYP3A4 (0.65) ALDH1A1HSD17B10TSHRCYP3A4CYP1A2
SCHEMBL561316 0.73 ADORA3 (0.64) ADORA3ALDH1A1HSD17B10HSP90AA1HSP90AB1
SCHEMBL28343462 0.72 CYP3A4 (0.69) ALDH1A1HSD17B10TSHRCYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0581500-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 1998-09-09 EP disclosed
US-5441949-A Carbapenem antibiotic compounds ZENECA LIMITED (GB) 1995-08-15 US disclosed
EP-0581500-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-02-02 EP disclosed