SCHEMBL8074189

SCHEMBL8074189

COC(=O)C1(c2ccc(OC)c(OC3CCCC3)c2)CCN(C(N)=O)C1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 20/20 0.59
PDE4A P27815 12/20 0.59
PDE4C Q08493 12/20 0.59
PDE4D Q08499 12/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7449841 0.88 PDE4B (0.64) PDE4BPDE4APDE4CPDE4D
SCHEMBL7445703 0.81 PDE4B (0.54) PDE4BPDE4APDE4CPDE4D
SCHEMBL7420740 0.74 PDE4A (0.66) PDE4BPDE4APDE4CPDE4D
SCHEMBL7416733 0.74 PDE4B (1.00) PDE4BPDE4APDE4CPDE4D
SCHEMBL7869812 0.74 PDE4B (0.76) PDE4BPDE4APDE4CPDE4D
SCHEMBL7375734 0.74 PDE4B (0.61) PDE4BPDE4APDE4CPDE4D
SCHEMBL6322995 0.73 PDE4B (0.74) PDE4BPDE4APDE4CPDE4D
SCHEMBL6323001 0.73 PDE4B (0.74) PDE4BPDE4APDE4CPDE4D
SCHEMBL6322447 0.73 PDE4B (0.74) PDE4BPDE4APDE4CPDE4D
SCHEMBL7443177 0.71 PDE4B (0.89) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0720600-B1 3-(3,4-DIOXYPHENYL)-PYRROLIDINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS FOR THE TREATMENT OF INFLAMMATORY DISEASES ICOS CORP (US) 2000-07-12 EP disclosed
US-5665754-A Substituted pyrrolidines GLAXO WELLCOME INC. (US) 1997-09-09 US disclosed