SCHEMBL807523

SCHEMBL807523

CC(C)c1c(Cl)cc(C#N)cc1C#N

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.34
AR P10275 4/20 0.34
ACACB O00763 1/20 0.33
TTR P02766 1/20 0.33
ALB P02768 1/20 0.33
VCAM1 P19320 2/20 0.32
CDK2 P24941 1/20 0.32
PGK1 P00558 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
GPR35 Q9HC97 1/20 0.30
KDM5A P29375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807269 0.87 TTR (0.38) ARTTRALBVCAM1ALDH1A1
SCHEMBL18552870 0.80 AR (0.39) ARTTRALBVCAM1KDM4E
SCHEMBL26457742 0.80 ALDH1A1 (0.35) TRPV4ARPGK1KDM4EALDH1A1
SCHEMBL13748821 0.78 AR (0.36) TRPV4ARPGK1ALDH1A1
SCHEMBL807272 0.78 MET (0.36) ARTTRALBVCAM1ALDH1A1
SCHEMBL15274595 0.78 ALDH1A1 (0.38) TRPV4ARPGK1KDM4EALDH1A1
SCHEMBL807520 0.78 TRPV4 (0.34) TRPV4TTRALBVCAM1
SCHEMBL13748310 0.76 AR (0.36) ARKDM4EALDH1A1
SCHEMBL13748825 0.76 PGR (0.34) TRPV4ARKDM5A
SCHEMBL15806352 0.75 AR (0.38) TRPV4ARTTRALBVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035039-A1 AZABENZOTHIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS OF USE F. HOFFMANN-LA ROCHE AG (CH) 2012-03-22 WO disclosed