SCHEMBL8075892

SCHEMBL8075892

Cc1cc(S(=O)(=O)Cl)c(C)cc1Cl.Cc1nc(-c2ccc(C(=O)N3CCN(S(=O)(=O)c4cc(C)c(Cl)cc4C)CC3)cc2)no1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.54
LMNA P02545 5/20 0.49
MAPT P10636 2/20 0.47
MGLL Q99685 2/20 0.47
CNR2 P34972 2/20 0.43
POLB P06746 1/20 0.43
ATM Q13315 1/20 0.43
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 2/20 0.42
HDAC4 P56524 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
CNR1 P21554 1/20 0.42
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7075338 0.96 THRB (0.58) THRBLMNAMAPTMGLLCNR2
SCHEMBL7074664 0.85 THRB (0.53) THRBLMNAMAPTMGLLATM
SCHEMBL7071363 0.84 MAPT (0.53) THRBLMNAMAPTMGLLALDH1A1
SCHEMBL7076931 0.82 MGLL (0.53) THRBLMNAMAPTMGLLALDH1A1
SCHEMBL8072947 0.81 THRB (0.46) THRBLMNAMGLLPOLBATM
SCHEMBL7069359 0.81 THRB (0.48) THRBLMNAMGLLATMALDH1A1
SCHEMBL7071746 0.81 MEN1 (0.54) LMNAMGLLPOLBALDH1A1KMT2A
SCHEMBL7076839 0.81 KMT2A (0.59) THRBLMNAMAPTMGLLPOLB
SCHEMBL7074158 0.80 MEN1 (0.68) THRBLMNAMAPTPOLBALDH1A1
SCHEMBL7074799 0.80 MGLL (0.55) THRBLMNAMGLLALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-A1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GmbH (DE) 2000-08-09 EP disclosed
WO-1999016751-A1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 1999-04-08 WO disclosed